BiologicalActivity
Potentvoltage-dependentNaV1.8channelblocker(IC50=11nMinrecombinanthumanNaV1.8channels).Reducestactileallodyniainneuropathicratmodels.3-and28-foldmorepotentatNaV1.8channelscomparedtoNaV1.2andNaV1.7channelsrespectively.
CompoundLibraries
A887826isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 480.99 |
| Formula | C26H29ClN4O3 |
| Storage | StoreatRT |
| Purity | ≥97%(HPLC) |
| CASNumber | 1266212-81-0 |
| PubChemID | 46919335 |
| InChIKey | JPJGFWKHSMUKFO-UHFFFAOYSA-N |
| Smiles | ClC1=C(OCCCC)C=CC(C2=CN=CC(C(NCC3=CC=CN=C3N4CCOCC4)=O)=C2)=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 24.05 | 50 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight480.99.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.08mL | 10.4mL | 20.79mL |
| 5mM | 0.42mL | 2.08mL | 4.16mL |
| 10mM | 0.21mL | 1.04mL | 2.08mL |
| 50mM | 0.04mL | 0.21mL | 0.42mL |
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