BiologicalActivity
PotentBRD9/7inhibitor(Kdvaluesare33and340nM,respectively)Exhibits>30-foldselectivityforBRD9overotherbromodomainsexceptBRD7.Cellpermeableandactiveinvivo.NegativecontrolTP472N(Cat.No.5999)available.
LicensingInformation
ThisprobeissuppliedinconjunctionwiththeStructuralGenomicsConsortium.Forfurthercharacterizationdetails,pleasevisittheTP472probesummaryontheSGCwebsite.
TechnicalData
| M.Wt | 333.38 |
| Formula | C20H19N3O2 |
| Storage | Storeat-20°C |
| Purity | ≥98%(HPLC) |
| PubChemID | 123773279 |
| InChIKey | RPBMXJHQYJLPDN-UHFFFAOYSA-N |
| Smiles | O=C(C)C1=CC(C2=CC(C(NC3CC3)=O)=CC=C2C)=C4N=CC=CN41 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 16.67 | 50 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight333.38.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 3mL | 15mL | 30mL |
| 5mM | 0.6mL | 3mL | 6mL |
| 10mM | 0.3mL | 1.5mL | 3mL |
| 50mM | 0.06mL | 0.3mL | 0.6mL |
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