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ubpbio/ONX-0914 (PR-957)/F1410/5 mg
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4000-520-616
ONX-0914,alsoknownasPR-957,isapotentinhibitoroftheimmunoproteasomewithminimalcross-reactivityfortheconstitutiveproteasome.ONX-0914selectivelyinhibitslow-molecularmasspolypeptide-7(LMP7),thesubunitspecificfortheimmunoproteasomethatcatalyzesthechymotyrpsion-likeactivity,withanIC50<100=""nm.=""cell=""culture=""and=""animal=""studies=""have=""shown=""that=""onx-0914=""blocks=""the=""production=""of=""proinflammatory=""cytokines=""including=""interleukin-6=""and=""17,=""indicating=""that=""it=""has=""potential=""uses=""in=""the=""treatment=""of=""some=""autoimmune=""diseases=""such=""as=""rheumatoid=""arthritis,=""inflammatory=""bowel=""disease=""and=""lupus.="">
Dose:0.1-0.5μMforinvitroorcellcoutureassays;intravenousorsubcutaneousadmiNISTrationat2-10mg/Kgdailyfor5-7daysforanimalstudies.
Dose:0.1-0.5μMforinvitroorcellcoutureassays;intravenousorsubcutaneousadmiNISTrationat2-10mg/Kgdailyfor5-7daysforanimalstudies.
AdditionalInformation
ProductName: | ONX-0914(PR-957) |
---|---|
AlsoKnownAs: | ONX0914;ONX0914;ONX-0914;PR-957;CAS#:960374-59-8 |
CatalogNo.: | F1410 |
Size: | 5mg |
MolecularWeight: | 580.7Da |
Species: | N/A |
Source: | Synthetic |
Stock: | Powder |
Concentration: | N/A |
QualityAssurance: | >98%byHPLCandNMR |
Storage: | EligIBLeforroomtemperatureshipping.Storeat-80°Cuponreceiving;avoidmultiplefreeze-thawcyclesafterdissolvinginDMSO. |
PDFDataSheet: | PDFDatasheet |
NCBIRefSeq: | N/A |
Image(s): | No |
ShippingMethod: | Roomtemperatureshipping |
References: | 1.MuchamuelT,etal.(2009)NatMed.15(7):781-7. 2.BaslerM,etal.(2010)JImmunol.185(1):634-41.3.KalimKW,etal.(2012)JImmunol.189(8):4182-93. |