BiologicalActivity
Potent,selectiveCysLT1(LTD4)leukotrienereceptorantagonist(IC50=6.4nM).InhibitsLTD4-inducedbronchoconstrictioninguineapigswhenadministeredintravenously,orallyorbyaerosol.
CompoundLibraries
CinalukastisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 412.55 |
| Formula | C23H28N2O3S |
| Storage | Desiccateat-20°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 128312-51-6 |
| PubChemID | 6436135 |
| InChIKey | BZMKNPGKXJAIDV-VAWYXSNFSA-N |
| Smiles | CCC(CC)(CC(=O)NC1=CC(C=CC2=NC(=CS2)C2CCC2)=CC=C1)C(O)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 41.26 | 100 | |
| ethanol | 4.13 | 10 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight412.55.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.42mL | 12.12mL | 24.24mL |
| 5mM | 0.48mL | 2.42mL | 4.85mL |
| 10mM | 0.24mL | 1.21mL | 2.42mL |
| 50mM | 0.05mL | 0.24mL | 0.48mL |
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