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Tocris/G-36/4759/50/50 mg
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Description:SelectiveGPERantagoNIST
ChemicalName:(±)-(3aR*,4S*,9bS*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-8-(1-methylethyl)-3H-cyclopenta[c]quinoline
Purity:≥99%(HPLC)
BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences
BiologicalActivity
AntagonistofGPER;selectivelyinhibitsestrogen-mediatedactivationofPI3-KbyGPER,butnotbyERα.Alsoinhibitsestrogen-mediatedcalciummobilization(IC50=112nM).StructuralanalogofG-1(Cat.No.3577).
TechnicalData
M.Wt | 412.33 |
Formula | C22H22BrNO2 |
Storage | Storeat-20°C |
Purity | ≥99%(HPLC) |
CASNumber | 1392487-51-2 |
PubChemID | 73755224 |
InChIKey | QTOCPACSSHFGOY-ZCCHDVMBSA-N |
Smiles | BrC1=CC4=C(OCO4)C=[C@@]1[C@@H]2NC(C=CC(C(C)C)=C5)=C5[C@@]3([H])[C@@]([H])2CC=C3 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
Solvent | MaxConc.mg/mL | MaxConc.mM | |
---|---|---|---|
Solubility | |||
DMSO | 41.23 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight412.33.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
---|---|---|---|
1mM | 2.43mL | 12.13mL | 24.25mL |
5mM | 0.49mL | 2.43mL | 4.85mL |
10mM | 0.24mL | 1.21mL | 2.43mL |
50mM | 0.05mL | 0.24mL | 0.49mL |
MolarityCalculator
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ReconstitutionCalculator
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DilutionCalculator
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ProductDatasheets
CertificateofAnalysis/ProductDatasheet
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