产品说明
CatalogNo.: B-0060MW: 405.46Purity: >98%CAS: 1345858-76-5Description: CYM50308isapotentandselectiveS1P4receptoragoNISTwithEC50of37.7nM-79.1nM.ItisinactiveagainsttheS1P1,S1P2,andS1P3receptorsupto25μM,andtheS1P5receptorupto2.1μM.Storage4°CReferences1)Urbanoetal.Discovery,synthesisandSARanalysisofnovelselectivesmallmoleculeS1P4-Ragonistsbasedona(2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-onechemotype,Bioorganic&MedicinalChemistryLetters,2011,6739-6745.2)Guerreroetal.Identificationofanovelagonistofthesphingosine1-phosphatereceptor4(S1P4),ProbeReportsfromtheNIHMolecularLibrariesProgram.http://www.ncbi.nlm.nih.gov/books/NBK143556/RelatedProductsSphingosineKinaseInhibitor(SK1-II)B-0024)2-Acetyl-5-tetrahydroxybutylimidazole(THI)(B-0031)NVP-231(CeramidekinaseInhibitor)(B-0040)FTY-720(B-0720)(S)-FTY720Phosphate(B-0721)
Echelon产品线
★合成磷脂、磷酸肌醇、鞘脂及其衍生物 |
★脂蛋白质相互作用工具 |
★脂质含量检测试剂盒 ★脂质相关生物酶活性检测,抑制剂筛选试剂盒 |
新品排行榜
1
Echelon/High Throughput Autotaxi...
2
Echelon/Tks5 VHH Antibody/250 ug...
3
Echelon/d5-D-myo-Phosphatidylino...
4
Echelon/Tensin 4 VHH Antibody/25...
5
Echelon/Autotaxin Inhibitor Scre...
6
Echelon/PTEN Activity ELISA Kit/...
7
Echelon/Hyaluronidase Activity E...
8
Echelon/Vinculin VHH Antibody/25...
9
Echelon/Vac14 Antibody, polyclon...
10
Echelon/Autotaxin Activity Assay...
文章排行榜
1
Echelon-inc
2
Echelon-inc
3
eBioscience AccutaseTM细胞分离溶液
4
eBioscience-莱兹生物免疫学技术讲座圆满落幕!
5
Echelon Bioscience公司简介,优势订购!
6
使用eBioscience流式抗体的常见问题
7
Echelon Biosciences 宣布与 ProBioscience Technologies 合作在东南亚分销 - Echelon Biosciences,Ebioscience 现货
8
FierceBiotech:2014年最热门的15家生物公司
9
Echelon Biosciences Incorporated中国采购 Echelon脂质含量检测试剂盒
10
Echelon经销商/代理商 Echelon抑制剂筛选试剂盒